Poster Session 2 — ASN Events

Poster Session 2 — ASN Events

Poster Session 2

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NanoBRET^TM assay for monitoring of ligand binding to GPCRs in live cells, using the CLARIOstar® and the PHERAstar® platereaders. (#136)

Spider toxin HwTx-IV engineered to bind to lipid membranes has an increased inhibitory potency at human voltage-gated sodium channel Na_V1.7 (#137)

Prediction of disulfide bond connectivity and configuration based on chemical shifts (#138)

David A Armstrong

Bioactive and stabilized cationic peptide capped metallic nanohybrid materials (#139)

Manish Mr. Bajaj

Novel capillary-flow LC HRAM MS platform for fast targeted analysis and robust profiling of complex samples (#140)

Using chemical methods to solve an antimicrobial engima (#141)

Silencing Intracellular Protein-Protein Interactions with Covalent Helical Peptide Inhibitors (#142)

Aline Dantas de Araujo

Harnessing structural conservation among serine proteases to engineer targeted inhibitors using a plant-derived cyclic peptide scaffold (#143)

Solution NMR characterisation of β-hairpin antimicrobial peptides in lipid bilayer nanodiscs. (#146)

Peptide-based antagonists of the Bcl-2-regulated apoptosis pathway (#147)

Improvement of oral delivery of EGFR-targeted hybrid peptide by combination with bile acid (#148)

Blm-pep based analogs with enhanced stimulatory capacity against human 20S proteasome (#149)

Malgorzata Gizynska

Elucidating the Rabies Virus P-protein Axis: Roles in Pathogenicity and Therapeutic Targeting (#150)

Design and Development of Selective AT2R Ligands (#152)

Synthesis and Structure Activity Relationship Studies of Insulin and Relaxin-like Peptides (#154)

Mohammed Akhter Hossain

Inhibitory effects of substrate-based BCR-ABL1 kinase inhibitors on drug-resistant chronic myeloid leukaemia cell lines (#155)

Phospholipid-mediated oligomerization of defensins induces fungal and tumour cell lysis (#156)

Structural and functional determinants for antimicrobial activity of sheep myeloid antimicrobial peptide-18 (SMAP-18) (#158)

Identification of a cyclotide antagonist at the corticotropin-releasing factor type 1 receptor (#159)

Synthesis of N^α -Fmoc-L-fluoroacetyl lysine for crosslinking of two functional groups in the context of close proximity provided by a peptide-protein complex (#160)

Marco Jan Klein

Stability tests of eye drops containing PACAP (#161)

Anita K. Kovacs

β‑peptide self-assembly as a new strategy for in situ bacterial detection and inhibition (#162)

Psd2 pea defensin’ preference for mimetic membranes rafts enriched with glucosylceramide and ergosterol (#164)

Eleonora Dr Kurtenbach

Development of novel relaxin-3 analogues for blood-brain barrier penetration (#166)

Proton conduction in a tyrosine-rich peptide/manganese oxide hybrid nanofilm (#167)

Global Analysis of O-GlcNAc Modification on alpha-Synuclein (#168)

Design and Synthesis of Xanthone-based Peptidomimetics as Antifungal Agents to Combat Fungal Resistance (#169)

Enhanced binding of the SOCS2 SH2-domain to phosphorylated targets by a novel exosite peptide (#170)

Understanding structure, self-assembly and biological activity of natural cyclic lipodepsipeptides by synthetic modification (#172)

Annemieke Madder

Identification of neuropeptide homologues in animal venoms using hidden markov models (#174)

Multivalent Ligand Design – Chemistry and Applications (#175)

Markus Muttenthaler

Peptide-based two-dimensional materials (#176)

Glycocin F: A glycosylated Cs α/α peptide with a novel antimicrobial activity (#177)

Peptide BDNF mimetics with central and peripheral nervous system actions (#178)

Susan E Northfield

Non-covalent sulfur-oxygen interactions control conformation in a peptidomimetic that disrupts islet amyloid polypeptide fibrillation (#181)

Hayden J Peacock

High throughput screening of large peptide libraries to identify drug specific formulation-additives or transporters (#182)

Polyunsaturated fatty acid-derived lipid mediators: their stability and detection in human plasma and the effect of a single dose of aspirin on their levels in healthy volunteers (#183)

Recombinant C-amidated antimicrobial peptide structural studies in whole bacteria using DNP solid-state NMR (#185)

Marc-Antoine Sani

Separation of complex peptide mixtures with displacement chromatography (#186)

Hartmut Schlueter

Targeted delivery of cyclotides via conjugation to a nanobody (#188)

Christina I Schroeder

Polymer-based peptide vaccine delivery systems. (#189)

Mariusz Skwarczynski

Ticks from Diverse Genera Encode Chemokine-Inhibitory Evasin Proteins (#191)

RaPID selection of macrocyclic peptides targeting ROR1 (#192)

Synthesis and characterisation of trefoil factor 3 loop mimetics (#193)

Synthesis and Functional Evaluation of Anti-Thrombotic Proteins Bearing Tyrosine Sulfation (#195)

Proteases in venom from jellyfish Nemopilema nomurai (#196)

Metalloantibiotics: old battles, new tricks. (#199)

A novel bifunctional chimera targeting both HIV-1 Env and host cell co-receptor (#200)

Biodistribution evaluation of ¹⁸⁸Re-liposome-SP90 in breast cancer solid tumor model (#201)

Liang-Cheng Chen

Identification and characterization of CHH-like neuropeptide receptors in the blackback land crab (Gecarcinus lateralis) molting gland transcriptome (#202)

Backbone cyclization of analgesic conotoxin GeXIVA facilitates direct folding of the ribbon isomer (#203)

Tracking and reporting synthetic peptide impurities with a cost-effective single quadrupole mass detector for improved confidence in analysis (#204)

Heather Patsiouras

Evaluation of a novel tandem quadrupole mass spectrometer for the multi-point internal calibration analysis of peptides (#205)

Heather Patsiouras

Enhancing vancomycin potency via complexation with silver ions (#206)

Hydroxylamine derivatives as new compounds to treat antibiotic bacterial resistance (#207)

Laia Miret Casals